Pregnant or planning a pregnancy? theophylline; If you are over 65 years of age, there may be specific risks and recommendations for use of this medicine. It is structurally similar to caffeine and is found in green and black tea. Find theophylline at best price offered by theophylline manufacturers, theophylline suppliers, dealers, traders and exporters. A methylxanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central nervous system stimulant activities. Nuelin SR Tablets contain 200 mg, 250 mg or 300 mg anhydrous theophylline in the form of sustained release tablets. As a member of the xanthine family, it bears structural and pharmacological similarity to theobromine and caffeine, and is readily found in nature, being present in tea and cocoa. Name Theophylline sodium glycinate Drug Entry Theophylline. Learn theophylline with free interactive flashcards. Provides a summary of interactions with vitamins, herbs, and food Theophylline. Choose from 124 different sets of theophylline flashcards on Quizlet. A blood test must be done to monitor your theophylline level to make sure the drug level is high enough to be effective, but not high enough to cause serious side effects. Additionally, it is essential that a patient discharged from hospital should be maintained on the brand on which that patient was stabilised as an in-patient. The most common side effects are headache, nausea and vomiting, abdominal discomfort, and restlessness. Send the page "" to a friend, relative, colleague or yourself. Email this page. “This is because the amount of theophylline absorbed by your body varies between brands,” says Dr Andy. https://www.cvs.com/drug/theophylline-anhydrous/oral-tablet-extended-release Theophylline is indicated for the-Control of acute asthma. USES: This medication is used to treat and prevent wheezing and trouble breathing caused by ongoing lung disease (e.g., asthma, emphysema, chronic bronchitis). This medication may be available under multiple brand names and/or in several different forms. Sticking to the same brand is important. From a pharmacokinetic point of view, doxofylline importantly differs from theophylline also because it lacks the ability to interfere with the cytochrome enzymes CYP1A2, CYP2E1 and CYP3A4, thus preventing significant interaction with other drugs metabolized via these pathways in the liver. There may also be … As theophylline (anhydrous) immediate-release solution: In patients who have not received theophylline or other xanthine agents in the previous 24 hours: Loading dose: 5 mg/kg to achieve an average of approx 10 mcg/mL peak serum levels. It can also be given intravenously (into a vein) for treatment for severe asthma attacks or COPD exacerbations. Measurement of plasma-theophylline concentration may be helpful and is essential if a loading dose of intravenous aminophylline is to be given to patients who are already taking theophylline, because serious side-effects such as convulsions and arrhythmias can occasionally precede other symptoms of toxicity. Your Name. Theophylline Theophylline is a bronchodilator that is not commonly used for COPD in the U.S. since most people can use inhaled bronchodilators. Theophylline belongs to a class of drugs known as xanthines. The pharmacokinetics of theophylline have been studied extensively in preterm neonates. Theophylline works by relaxing the smooth muscles of the airways while relieving inflammation and a… Management of chronic obstructive lung disease (Chronic bronchitis and emphysema) and acute exacerbation of chronic … FILTER BY COMPANY ACI Limited ACME … Theophylline is sold as a generic pill or under the brand names Theo-24 and Uniphyl. It also has mild diuretic effects. Theophylline, an xanthine derivative chemically similar to caffeine and theobromine, is used to treat asthma and bronchospasm. Dosage requirement must be guided by the patient’s serum theophylline concentrations, safety, and tolerability (refer to detailed product guideline). Do I need a prescription for theophylline? If a prescription for an oral theophylline MR preparation does not specify a brand name, the pharmacist should contact the Due to its numerous side-effects, these drugs are now rarely administered for clinical use. Elixophyllin, Theo-24. What is theophylline? Retrouvez sur VIDAL la liste des médicaments contenant la substance active Théophylline : DILATRANE, EUPHYLLINE L.A. A small … Thus, drugs that inhibit CYP1A2, such as macrolide and quinolone antibiotics, cimetidine, and fluvoxamine, may increase plasma theophylline concentrations to levels that produce side effects. Theophylline View all Brand Names Innovator's Monograph Indications. Theophylline is a dimethylxanthine having the two methyl groups located at positions 1 and 3. It’s available as an oral (pill and liquid) or intravenous (through the vein) drug. Please discuss your individual circumstances with your pharmacist, doctor or health professional. Theophylline is a safe, effective drug for the treatment of apnea of prematurity. Mechanistically, theophylline acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator. oral, IV. Make sure you get the same brand of theophylline each time you pick up a new prescription. Nuelin SR Tablets also contain guar gum, magnesium stearate and purified water. Message. Brand Names and Other Names of Theophylline; This drug is registered for use in humans only. For more information read our page on medication safety for older people. Get information of companies selling wide range of theophylline along with latest price, moq & product details. BRAND NAME(S): Uniphyl. Theophylline has two distinct actions in the airways of patients with reversible (asthmatic) obstruction; smooth muscle relaxation (i.e., bronchodilation) and suppression of the response of the airways to stimuli (i.e., non-bronchodilator prophylactic effects). Theophylline helps to ease the cough, wheezing, shortness of breath, and troubled breathing associated with these conditions by allowing relaxation of the tubes (bronchi) of the airways, thereby permitting increased amounts of air to flow through them. Theophylline is metabolized in the liver by the P-450 isoenzyme CYP1A2 . Is theophylline available as a generic drug? Theophylline, also known as dimethylxanthine, is a methylxanthine drug used in therapy for respiratory diseases such as COPD or asthma under a variety of brand names. For the active ingredient theophylline. ChEBI Name theophylline: ChEBI ID CHEBI:28177: Definition A dimethylxanthine having the two methyl groups located at positions 1 and 3. If a prescription for a modified-release oral theophylline preparation does not specify a brand name, the pharmacist should contact the prescriber and agree the brand to be dispensed. It is structurally similar to caffeine and is … Management of chronic asthma (For both Symptomatic and prophylactic treatment). It is usually taken by mouth as a pill. Nuelin Syrup contains 133.3 mg anhydrous theophylline per 25 mL in immediate release form. 1981 Oct;5(4):337-45. The molecular formula of anhydrous theophylline is C 7 H 8 N 4 O 2 with a molecular weight of 180.17.. Theo-24 (theophylline anhydrous capsule) ® is available as capsules intended for oral administration, containing 100 mg, 200 mg, 300 mg, or 400 mg of anhydrous theophylline per capsule, in an extended-release formulation which allows a 24-hour dosing interval for appropriate patients. Theophylline is considered a component of a treatment plan. It is typically taken by mouth for the long-term control and maintenance of asthma, COPD (including emphysema and chronic bronchitis), and other chronic lung diseases. Yes. Theophylline Available Brands. What brand names are available for theophylline? Required field. Human formulations: Theo-Dur® (Key Pharmaceuticals) and various generic brands are available. Theophylline is marketed under several brand names such as Uniphyl and Theochron, and it is indicated mainly for asthma, bronchospasm, and COPD. Aminophylline is monitored therapeutically in terms of plasma-theophylline concentrations. Some are considered “extended release” preparations, exhibiting a longer duration of effect. Patients should be maintained on the same brand [4, 17 ]. Separate multiple email address with a comma. It has a role as a vasodilator agent, a bronchodilator agent, a muscle relaxant, an EC 3.1.4. For controlling nocturnal asthma and early morning wheezing. Theophylline MR preparations Theophylline has a narrow therapeutic index and bioavailability differs between brands of oral MR theophylline. Yes. Theophylline, also known as 1,3-dimethylxanthine, is a phosphodiesterase inhibiting drug used in therapy for respiratory diseases such as chronic obstructive pulmonary disease and asthma under a variety of brand names. Theophylline is used for the relief and prevention of airway narrowing (bronchospasm) in patients with asthma. Recipient's Email. (a) You are authorized to use the AAP’s trademarks, logos and brand names (the “ AAP Trademarks ”) only in connection with reproducing any such AAP Trademarks as incorporated in the Materials. Home / Theophylline Extended-Release Tablets (100 mg, 200 mg, 300 mg, 450 mg) Drug Information / Drug Summary email print Close window. Medication Uses | How To Use | Side Effects | Precautions | Drug Interactions | Overdose | Notes | Missed Dose | Storage. Drug Name : Theophylline Theophylline (Aquaphyllin) generic is a bronchodilator, prescribed for asthma, chronic bronchitis, emphysema, and other lung diseases. Mechanistically, theophylline acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator. What are the uses for theophylline? Names There is some inter-infant variability, but generally, compared to children and adults, prolonged half-life values and low clearan … Pharmacokinetics of theophylline in neonates Semin Perinatol. Its use in cats and dogs to treat cough and bronchoconstriction is 'off label' or 'extra label.Many drugs are commonly prescribed for off label use in veterinary medicine. P (UK) Routes. 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